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Modiodal Modafinil

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Modiodal Modafinil
#1
Le modafinil est également un inhibiteur de la recapture de la noradrénaline. D'autres facteurs peuvent également influencer la façon dont le modafinil interagit avec vos autres médicaments, vous devez donc en parler à votre médecin. Le modafinil est un activateur dopaminergique. Dans le même temps, les antipsychotiques atypiques semblent bloquer les propriétés d'amélioration de l'éveil du modafinil. Le modafinil est utilisé comme activateur cognitif pour améliorer l'éveil. Le modafinil est généralement administré par voie orale sous forme de comprimés et généralement pris au moment d'un épisode de sommeil (vraisemblablement au coucher). Modiodal Modafinil Il n'a pas été étudié à d'autres fins, y compris le trouble déficitaire de l'attention (ADD) et le trouble déficitaire de l'attention avec hyperactivité (TDAH). Bien que le modafinil soit approuvé pour l'utilisation à court terme de la narcolepsie et de l'apnée du sommeil, son innocuité pendant la grossesse est inconnue. Le modafinil agit sur des parties du cerveau qui régulent les rythmes circadiens, lui permettant d'exercer ses effets tout au long du cycle veille-sommeil. La dose initiale recommandée de modafinil est de 100 mg une fois par jour et la dose peut être augmentée par paliers de 100 mg jusqu'à un maximum de 600 mg par jour. Aucune réaction cardiovasculaire grave n'a été signalée dans les essais cliniques, bien qu'elle ait provoqué une surstimulation chez quelques personnes. Plus précisément, le modafinil a été qualifié d'"agoniste α2", ce qui signifie qu'il s'agit d'un agoniste faible du récepteur alpha-2. Certaines personnes peuvent bénéficier du modafinil et cela dépend si leur corps métabolise le modafinil différemment. Le modafinil est principalement métabolisé par l'enzyme hépatique CYP3A4. Lorsque Modafinil est ingéré, il pénètre dans le système nerveux central en traversant la barrière hémato-encéphalique. Il est utilisé pour traiter certains cas de narcolepsie et de troubles du sommeil liés au travail posté. Alors que le modafinil est recommandé à 100 mg pour les personnes souffrant de troubles du sommeil liés au travail posté ou à 200 mg pour les personnes atteintes de narcolepsie, les doses sont extrapolées à partir d'études avec d'autres indications et peuvent être ajustées. Le nom chimique du modafinil est le chlorhydrate de 1-[(diphénylméthyl)sulfinyl]-2-[4-(méthylthio)phényl]méthoxyéthan-1-amine. Le modafinil peut également être utile pour une variété d'autres conditions. Le modafinil (Provigil) est un stimulant du système nerveux central utilisé pour traiter la somnolence associée à la narcolepsie, les troubles du sommeil liés au travail posté et l'apnée obstructive du sommeil. Le modafinil est une «substance activatrice» qui affecte le noyau tegmental dorsal du pont.

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